Recent developments of carbonic anhydrase inhibitors as potential drugs

Recent developments of carbonic anhydrase inhibitors as potential drugs (151 visite)

Iqbal J, Al-rashida M, Durdagi S, Alterio V, Di Fiore A

Biomed Res Int (ISSN: 2314-6133, 2314-6141), 2015; 2015: 174178-174178.

Tipo di articolo: Journal Article, Editorial, Introductory Journal Article,

Impact factor: 2.134, Impact factor a 5 anni: 2.149

Url: http://www.scopus.com/inward/record.url?eid=2-s2.0-84925340753&partnerID=40&md5=388ebd0c931495d70b27bbd4f9780166

Parole chiave: Carbonate Dehydratase, Carbonate Dehydratase Ii, Carbonate Dehydratase Inhibitor, Carbonate Dehydratase Vii, Carbonate Dehydratase Xii, Exportin 1, Polyamine Derivative, Saccharin Derivative, Spermidine, Sulfanilamide Derivative, Unclassified Drug, Catalysis, Crystal Structure, Disorders Of Acid Base Balance, Editorial, Enzyme Inhibition, Epilepsy, Glaucoma, Neoplasm, Nonhuman, Obesity, Stomach Ulcer, Binding Sites, Carbonic Anhydrase Inhibitors, Chemical Synthesis, Chemistry, Ultrastructure, Drug Design, Enzyme Activation, Drug Effects, Enzyme Stability, Protein Binding,

Affiliazioni:

*** IBB - CNR ***
Department of Pharmaceutical Sciences, Centre for Advanced Drug Research, COMSATS Institute of Information Technology, Abbottabad, Pakistan
Department of Chemistry, Forman Christian College, A Chartered University, Ferozepur Road, Lahore, Pakistan
Department of Basic Medical Sciences, School of Medicine, Bahçeşehir University, Turkey
Institute of Biostructure and Bioimaging (IBB), Italian National Research Council, Via Mezzocannone 16, Naples, Italy

Riferimenti:

Non disponibile.

Non disponibile.

Interrogazione effettuata: [atitle, keywords] "Carbonate Dehydratase" OR [atitle, keywords] "Carbonate Dehydratase Ii" OR [atitle, keywords] "Carbonate Dehydratase Inhibitor" OR [atitle, keywords] "Carbonate Dehydratase Vii" OR [atitle, keywords] "Carbonate Dehydratase Xii" OR [atitle, keywords] "Exportin 1" OR [atitle, keywords] "Polyamine Derivative"

Nessun risultato.

Interrogazione effettuata: [ptitle] "Carbonate Dehydratase" OR [ptitle] "Carbonate Dehydratase Ii" OR [ptitle] "Carbonate Dehydratase Inhibitor" OR [ptitle] "Carbonate Dehydratase Vii" OR [ptitle] "Carbonate Dehydratase Xii" OR [ptitle] "Exportin 1" OR [ptitle] "Polyamine Derivative"

Nessun risultato.

Interrogazione effettuata: [btitle, keywords] "Carbonate Dehydratase" [btitle, keywords] "Carbonate Dehydratase Ii" [btitle, keywords] "Carbonate Dehydratase Inhibitor" [btitle, keywords] "Carbonate Dehydratase Vii" [btitle, keywords] "Carbonate Dehydratase Xii" [btitle, keywords] "Exportin 1" [btitle, keywords] "Polyamine Derivative"

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Calabrese V, Mancuso C, Calvani M, Rizzarelli E, Butterfield DA, Stella AM
* Nitric oxide in the central nervous system: neuroprotection versus neurotoxicity (242 visite)
Nature Reviews Neuroscience (ISSN: 1471-0048), 2007 Oct; 8(10): 766-775.
Impact Factor: 24.52
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Alterio V, De Simone G, Monti SM, Scozzafava A, Supuran CT
* Carbonic anhydrase inhibitors: Inhibition of human, bacterial, and archaeal isozymes with benzene-1, 3-disulfonamides-Solution and crystallographic studies (138 visite)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x), 2007 Sep 1; 17(15): 4201-4207.
Impact Factor: 2.604
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Vitale RM, Pedone C, Amodeo P, Antel J, Wurl M, Scozzafava A, Supuran CT, De Simone G
* Molecular modeling study for the binding of zonisamide and topiramate to the human mitochondrial carbonic anhydrase isoform VA (138 visite)
Bioorg Med Chem (ISSN: 0968-0896, 1464-3391, 1464-3391electronic), 2007 Jun 15; 15(12): 4152-4158.
Impact Factor: 2.662
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Di Fiore A, Scozzafava A, Winum JY, Montero JL, Pedone C, Supuran CT, De Simone G
* Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties (140 visite)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x), 2007 Mar 15; 17(6): 1726-1731.
Impact Factor: 2.604
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Ronga L, Palladino P, Costantini S, Facchiano A, Ruvo M, Benedetti E, Ragone R, Rossi F
* Conformational diseases and structure-toxicity relationships: Lessons from prion-derived peptides (194 visite)
Curr Protein Pept Sci (ISSN: 1389-2037), 2007 Feb; 8(1): 83-90.
Impact Factor: 3.259
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De Simone G, Supuran CT
* Antiobesity carbonic anhydrase inhibitors (179 visite)
Curr Top Med Chem (ISSN: 1568-0266, 1568-0266linking, 1873-4294electronic), 2007; 7(9): 879-884.
Impact Factor: 4.325
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Leese MP, Leblond B, Smith A, Newman SP, Di Fiore A, De Simone G, Supuran CT, Purohit A, Reed MJ, Potter BVL
* 2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity (327 visite)
J Med Chem (ISSN: 0022-2623print, 0022-2623linking, 1520-4804), 2006 Dec 28; 49(26): 7683-7696.
Impact Factor: 5.115
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Menchise V, De Simone G, Di Fiore A, Scozzafava A, Supuran CT
* Carbonic anhydrase inhibitors: X-ray crystallographic studies for the binding of 5-amino-1, 3, 4-thiadiazole-2-sulfonamide and 5-(4-amino-3-chloro-5-fluorophenylsulfonamido)1, 3, 4-thiadiazole-2-sulfon amide to human isoform II (123 visite)
Bioorganic & Medicinal Chemistry Letters (ISSN: 0960-894x), 2006 Dec 15; 16(24): 6204-6208.
Impact Factor: 2.538
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De Simone G, Vitale RM, Di Fiore A, Pedone C, Scozzafava A, Montero JL, Winum JY, Supuran CT
* Carbonic anhydrase inhibitors: Hypoxia-activatable sulfonamides incorporating disulfide bonds that target the tumor-associated isoform IX (160 visite)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print), 2006 Sep 7; 49(18): 5544-5551.
Impact Factor: 5.115
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Alterio V, Vitale RM, Monti SM, Pedone C, Scozzafava A, Cecchi A, De Simone G, Supuran CT
* Carbonic anhydrase inhibitors: X-ray and molecular modeling study for the interaction of a fluorescent antitumor sulfonamide with isozyme II and IX (135 visite)
J Am Chem Soc (ISSN: 0002-7863, 0002-2786, 1520-5126), 2006 Jun 28; 128(25): 8329-8335.
Impact Factor: 7.696
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Di Fiore A, Pedone C, D'Ambrosio K, Scozzafava A, De Simone G, Supuran CT
* Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II 'selective' inhibitor celecoxib (137 visite)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x), 2006 Jan 15; 16(2): 437-442.
Impact Factor: 2.538
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Menchise V, De Simone G, Alterio V, Di Fiore A, Pedone C, Scozzafava A, Supuran CT
* Carbonic anhydrase inhibitors: Stacking with Phe131 determines active site binding region of inhibitors as exemplified by the X-ray crystal structure of a membrane-impermeant antitumor sulfonamide complexed with isozyme II (172 visite)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print), 2005 Sep 8; 48(18): 5721-5727.
Impact Factor: 4.926
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De Simone G, Di Fiore A, Menchise V, Pedone C, Antel J, Casini A, Scozzafava A, Wurl M, Supuran CT
* Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies (131 visite)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x), 2005 May 2; 15(9): 2315-2320.
Impact Factor: 2.478
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Di Fiore A, De Simone G, Menchise V, Pedone C, Casini A, Scozzafava A, Supuran CT
* Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II (167 visite)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x), 2005 Apr 1; 15(7): 1937-1942.
Impact Factor: 2.478
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Fonti R, Latella G, Caprilli R, Frieri G, Marcheggiano A, Sambuy Y
Carbonic anhydrase I reduction in colonic mucosa of patients with active ulcerative colitis (91 visite)
Digestive Diseases And Sciences (ISSN: 0163-2116), 1998; 43(9): 2086-2092.
Impact Factor: 1.972
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70 Records (69 escludendo Abstract e Conferenze).
Impact factor totale: 368.156 (363.041 escludendo Abstract e Conferenze).
Impact factor a 5 anni totale: 370.763 (365.259 escludendo Abstract e Conferenze).

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