Carbonic Anhydrases: An Overview
Menu piccolo
Institute
About us
Documents
News
Organization chart
Locations
Staff
Contact us
Activities
Education
Career opportunities
Meetings
PNRR
Research
Research Areas
Biomolecules
Imaging
e-Health
Projects
Publications
Patents
Resources
Awards and acknowledgments
Statistics
Private Area
Login
Link utili
Staff
Research areas
Activities
Bibliography
Papers
CMS
Generic
IT
Basic info
Abstract
Related activities
Related bibliography
Carbonic Anhydrases: An Overview
(
395 views
)
Supuran CT,
De Simone G
Carbonic Anhydrases As Biocatalysts
,
2015 Jan 08;
N/D: 3-13.
Export to BibTeX
Export to EndNote
Paper type:
Book Chapter,
Impact factor:
0,
5-year impact factor:
0
Url:
Not available.
Keywords:
Not available.
Affiliations:
Not available.
References:
Not available.
Carbonic Anhydrases: An Overview
Not available.
Carbonic Anhydrases: An Overview
▼
Carbonic Anhydrase family as target for rational drug design
Monti Simona Maria
De Simone Giuseppina
Alterio Vincenzo
▼
Carbonic Anhydrase IX as target for the development of new anti-tumour drugs
Buonanno Martina
Monti Simona Maria
Langella Emma
Di Fiore Anna
D'Ambrosio Katia
De Simone Giuseppina
Alterio Vincenzo
Carbonic Anhydrases: An Overview
Filter those results▼
Query: [
X
]
Options:
Any
All
Exact
Extended
IBB affiliation
OR
AND
Authors: [
X
]
Paper type: [
X
]
Start date: [
X
]
End date: [
X
]
Site:
All sites
Naples - De Amicis
Naples - Castellino
Turin
Staff
Research areas
Activities
Bibliography
Papers
CMS
Generic
[
Clear form
]
Select the year:
Default
ALL YEARS
2025
2024
2023
2022
2021
2020
2019
2018
2017
2016
2015
2014
2013
2012
2011
2010
2009
2008
2007
2006
2005
2004
2003
2002
<=2001
Other filter:
([btitle,keywords] "Carbonic" OR [btitle ...
Search related bibliography on PubMed
End of page
Copy&Paste Friendly
Export all to BibTeX
Export all to EndNote
Sort by: date
▼
▲
title
▲
▼
journal
▲
▼
authors
▲
▼
I.F.
▲
▼
Nocentini A, Bonardi A, Bazzicalupi C,
Alterio V
,
Esposito D
,
Monti SM
, Smietana M,
De Simone G
, Supuran CT, Gratteri P, Winum JY
*
6-Substituted Triazolyl Benzoxaboroles as Selective Carbonic Anhydrase Inhibitors: In Silico Design, Synthesis, and X-ray Crystallography
(
124 views
)
J Med Chem (ISSN: 0022-2623linking)
,
2023 Jun 22;
66 (12 ): 8118-8129.
Impact Factor:
View
Export to BibTeX
Export to EndNote
Langella E
,
Esposito D
,
Monti SM
, Supuran CT,
De Simone G
,
Alterio V
*
A Combined in Silico and Structural Study Opens New Perspectives on Aliphatic Sulfonamides, a Still Poorly Investigated Class of CA Inhibitors
(
187 views
)
Biology (ISSN: 2079-7737linking)
,
2023 Feb 10;
12 (2 ): N/D-N/D.
Impact Factor:
View
Export to BibTeX
Export to EndNote
Di Fiore A
, De Luca V,
Langella E
, Nocentini A,
Buonanno M
,
Monti SM
, Supuran CT, Capasso C,
De Simone G
*
Biochemical, structural, and computational studies of a γ-carbonic anhydrase from the pathogenic bacterium Burkholderia pseudomallei
(
100 views
)
Comput Struct Biotechnol J (ISSN: 2001-0370linking)
,
2022 Jul 27;
20: 4185-4194.
Impact Factor:
6.155
View
Export to BibTeX
Export to EndNote
Sarnella A
,
Ferrara Y
,
Auletta L
,
Albanese S
, Cerchia L,
Alterio V
,
De Simone G
, Supuran CT,
Zannetti A
*
Inhibition of carbonic anhydrases IX/XII by SLC-0111 boosts cisplatin effects in hampering head and neck squamous carcinoma cell growth and invasion
(
132 views
)
J Exp Clin Canc Res (ISSN: 0392-9078linking, 1756-9966, 1756-9966electronic)
,
2022 Apr 2;
41(1): 122-122.
Impact Factor:
12.658
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Supuran CT, Scaloni A,
De Simone G
*
Post-translational modifications in tumor-associated carbonic anhydrases
(
141 views
)
Amino Acids (ISSN: 0939-4451linking, 1438-2199electronic)
,
2022 Apr;
54(4): 543-558.
Impact Factor:
3.46
View
Export to BibTeX
Export to EndNote
Akgül Ö, Lucarini E, Mannelli LDC, Ghelardini C, D'Xambrosio K,
Buonanno M
,
Monti SM
,
De Simone G
, Angeli A, Supuran CT, Carta F
*
Sultam based Carbonic Anhydrase VII inhibitors for the management of neuropathic pain
(
104 views
)
Eur J Med Chem (ISSN: 0223-5234linking, 1768-3254, 1768-3254electronic)
,
2022 Jan 5;
227: 113956-113956.
Impact Factor:
7.088
View
Export to BibTeX
Export to EndNote
Pagnozzi D, Pala N, Biosa G, Dallocchio R, Dessì A, Singh PK, Rogolino D,
Di Fiore A
,
De Simone G
, Supuran CT, Sechi M
*
Interaction Studies between Carbonic Anhydrase and a Sulfonamide Inhibitor by Experimental and Theoretical Approaches
(
140 views
)
Acs Med Chem Lett
,
2022;
13: 271-277.
Impact Factor:
4.632
View
Export to BibTeX
Export to EndNote
Urbański LJ, Angeli A, Hytönen VP,
Di Fiore A
,
De Simone G
, Parkkila S, Supuran CT
*
Inhibition of the β-carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with sulphonamides
(
228 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366linking, 1475-6374electronic)
,
2021 Dec;
36(1): 329-334.
Impact Factor:
4.673
View
Export to BibTeX
Export to EndNote
Troisi R, Balasco N,
Autiero I
,
Vitagliano L
,
Sica F
*
Exosite Binding in Thrombin: A Global Structural/Dynamic Overview of Complexes with Aptamers and Other Ligands
(
123 views
)
Int J Mol Sc (ISSN: 1422-0067linking, 1422-0067electronic, 1661-6596)
,
2021 Oct 6;
22 (19 ): N/D-N/D.
Impact Factor:
2.598
View
Export to BibTeX
Export to EndNote
Del Gatto A
, Saviano M,
Zaccaro L
*
An Overview of Peptide-Based Molecules as Potential Drug Candidates for Multiple Sclerosis
(
137 views
)
Molecules (ISSN: 1420-3049linking, 1420-3049electronic)
,
2021 Aug 28;
26(17): N/D-N/D.
Impact Factor:
4.411
View
Export to BibTeX
Export to EndNote
Mancuso F,
Di Fiore A
,
De Luca L
, Angeli A,
De Simone G
, Supuran CT, Gitto R
*
Design, synthesis and biochemical evaluation of novel carbonic anhydrase inhibitors triggered by structural knowledge on hCA VII
(
164 views
)
Bioorg Med Chem (ISSN: 0968-0896linking, 1464-3391)
,
2021 Aug 15;
44: 116279-116279.
Impact Factor:
3.641
View
Export to BibTeX
Export to EndNote
Alterio V
,
Langella E
,
Buonanno M
,
Esposito D
, Nocentini A, Berrino E, Bua S, Polentarutti M, Supuran CT,
Monti SM
,
De Simone G
*
Zeta-carbonic anhydrases show CS(2) hydrolase activity: A new metabolic carbon acquisition pathway in diatoms?
(
179 views
)
Comput Struct Biotechnol J (ISSN: 2001-0370linking)
,
2021 Jun 5;
19: 3427-3436.
Impact Factor:
7.271
View
Export to BibTeX
Export to EndNote
De Simone G
, Bua S, Supuran CT,
Alterio V
*
Benzyl alcohol inhibits carbonic anhydrases by anchoring to the zinc coordinated water molecule
(
125 views
)
Biochem Biophys Res Commun (ISSN: 0006-291xlinking)
,
2021 Apr 9;
548: 217-221.
Impact Factor:
3.575
View
Export to BibTeX
Export to EndNote
Vincenzi M,
Mercurio FA
,
Leone M
*
NMR spectroscopy in the conformational analysis of peptides: an overview
(
200 views
)
Curr Med Chem (ISSN: 0929-8673linking, 1875-533xelectronic)
,
2021;
28(14): 2729-2782.
Impact Factor:
4.184
View
Export to BibTeX
Export to EndNote
D’ambrosio K,
Di Fiore A
,
Buonanno M
, Kumari S, Tiwari M, Supuran CT, Mishra CB,
Monti SM
,
De Simone G
*
The crystal structures of 2-(4-benzhydrylpiperazin-1-yl)-N-(4-sulfamoylphenyl)acetamide in complex with human carbonic anhydrase II and VII provide insights into selective CA inhibitor development
(
171 views
)
New Journal Of Chemistry
,
2021;
45: 147-152.
Impact Factor:
3.288
View
Export to BibTeX
Export to EndNote
Squeglia F
,
Romano M
,
Ruggiero A
, Maga G,
Berisio R
*
Host DDX Helicases as Possible SARS-CoV-2 Proviral Factors: A Structural Overview of Their Hijacking Through Multiple Viral Proteins
(
198 views
)
Front Chem (ISSN: 2296-2646linking)
,
2020 Dec 10;
8: 602162-602162.
Impact Factor:
3.693
View
Export to BibTeX
Export to EndNote
Spagnuolo R, Abenavoli L, Larussa T, Iannelli C, Pellicano R,
Fagoonee S
, Doldo P, Luzza F
*
Safety profile of intravenous iron in inflammatory bowel disease: an up-to-date overview
(
313 views
)
Minerva Gastroenterol Dietol (ISSN: 1121-421xlinking)
,
2020 Dec 3;
N/D: N/D-N/D.
Impact Factor:
2.36
View
Export to BibTeX
Export to EndNote
Urbański LJ,
Di Fiore A
, Azizi L, Hytönen VP, Kuuslahti M,
Buonanno M
,
Monti SM
, Angeli A, Zolfaghari Emameh R, Supuran CT,
De Simone G
, Parkkila S
*
Biochemical and structural characterisation of a protozoan beta-carbonic anhydrase from Trichomonas vaginalis
(
216 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366linking, 1475-6374electronic)
,
2020 Dec;
35(1): 1292-1299.
Impact Factor:
4.673
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Supuran CT, Scaloni A,
De Simone G
*
Human carbonic anhydrases and post-translational modifications: a hidden world possibly affecting protein properties and functions
(
243 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366linking, 1475-6374electronic)
,
2020 Dec;
35(1): 1450-1461.
Impact Factor:
4.673
View
Export to BibTeX
Export to EndNote
Urbański LJ, Angeli A, Hytönen VP,
Di Fiore A
, Parkkila S,
De Simone G
, Supuran CT
*
Inhibition of the newly discovered β‑carbonic anhydrase from the protozoan pathogen Trichomonas vaginalis with inorganic anions and small molecules
(
190 views
)
J Chem Res (ISSN: 0162-0134linking, 0162-0134print, 1873-3344)
,
2020 Dec;
213: 111274-111274.
Impact Factor:
3.212
View
Export to BibTeX
Export to EndNote
Sarnella A
, D'Avino G, Hill BS,
Alterio V
, Winum JY, Supuran CT,
De Simone G
,
Zannetti A
*
A Novel Inhibitor of Carbonic Anhydrases Prevents Hypoxia-Induced TNBC Cell Plasticity
(
190 views
)
(PDF
52 views
)
Int J Mol Sc (ISSN: 1422-0067linking, 1422-0067electronic, 1661-6596)
,
2020 Nov 9;
21(21): N/D-N/D.
Impact Factor:
4.556
View
Export to BibTeX
Export to EndNote
D'Ambrosio K
, Carradori S, Cesa S, Angeli A,
Monti SM
, Supuran CT,
De Simone G
*
Catechols: a new class of carbonic anhydrase inhibitors
(
139 views
)
Chem Commun (ISSN: 1359-7345linking, 1364-548xelectronic)
,
2020 Nov 4;
56(85): 13033-13033.
Impact Factor:
5.996
View
Export to BibTeX
Export to EndNote
Angeli A, Carta F, Nocentini A, Winum J, Zalubovskis R, Akdemir A, Onnis V, Eldehna WM, Capasso C,
De Simone G
, Monti Simona M, Carradori S, Donald WA, Dedhar S, Supuran CT
*
Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment
(
188 views
)
Metabolites
,
2020 Oct 14;
10: 412-412.
Impact Factor:
4.097
View
Export to BibTeX
Export to EndNote
Bozdag M, Supuran CT,
Esposito D
, Angeli A, Carta F,
Monti SM
,
De Simone G
,
Alterio V
*
2-Mercaptobenzoxazoles: a class of carbonic anhydrase inhibitors with a novel binding mode to the enzyme active site
(
170 views
)
Chem Commun (ISSN: 1359-7345linking, 1364-548xelectronic)
,
2020 Jul 23;
56(59): 8297-8300.
Impact Factor:
5.996
View
Export to BibTeX
Export to EndNote
Nocentini A,
Alterio V
, Bua S, Micheli L,
Esposito D
,
Buonanno M
, Bartolucci G, Osman SM, Alothman ZA, Cirilli R, Pierini M,
Monti SM
, Di Cesare Mannelli L, Gratteri P, Ghelardini C,
De Simone G
, Supuran CT
*
Phenyl(thio)phosphon(amid)ate Benzenesulfonamides as Potent and Selective Inhibitors of Human Carbonic Anhydrases II and VII Counteract Allodynia in a Mouse Model of Oxaliplatin-Induced Neuropathy
(
257 views
)
J Med Chem (ISSN: 0022-2623linking, 0022-2623print, 1520-4804)
,
2020 May 28;
63(10): 5185-5200.
Impact Factor:
6.205
View
Export to BibTeX
Export to EndNote
Mancuso F,
Di Fiore A
,
De Luca L
, Angeli A,
Monti SM
,
De Simone G
, Supuran CT, Gitto R
*
Looking toward the Rim of the Active Site Cavity of Druggable Human Carbonic Anhydrase Isoforms
(
259 views
)
Acs Med Chem Lett (ISSN: 1948-5875linking)
,
2020 May 14;
11(5): 1000-1005.
Impact Factor:
3.975
View
Export to BibTeX
Export to EndNote
Langella E
,
Buonanno M
,
De Simone G
,
Monti SM
*
Intrinsically disordered features of carbonic anhydrase IX proteoglycan-like domain
(
170 views
)
Cell Mol Life Sci (ISSN: 1420-682xlinking)
,
2020;
21: 8405-8405.
Impact Factor:
6.496
View
Export to BibTeX
Export to EndNote
Alterio V
, Kellner M,
Esposito D
, Liesche-starnecker F, Bua S, Supuran CT,
Monti SM
, Zeidler R,
De Simone G
*
Biochemical and structural insights into Carbonic Anhydrase XII/Fab6A10 complex
(
239 views
)
J Mol Biol (ISSN: 0022-2836linking, 1089-8638)
,
2019 Dec 6;
431(24): 4910-4921.
Impact Factor:
5.067
View
Export to BibTeX
Export to EndNote
De Simone G
,
Di Fiore A
, Truppo E,
Langella E
, Vullo D, Supuran CT,
Monti SM
*
Exploration of the residues modulating the catalytic features of human carbonic anhydrase XIII by a site-specific mutagenesis approach
(
328 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366linking, 1475-6374electronic)
,
2019 Dec;
34(1): 1506-1510.
Impact Factor:
4.027
View
Export to BibTeX
Export to EndNote
Langella E
,
Alterio V
,
D'Ambrosio K
, Cadoni R, Winum JY, Supuran CT,
Monti SM
,
De Simone G
,
Di Fiore A
*
Exploring benzoxaborole derivatives as carbonic anhydrase inhibitors: a structural and computational analysis reveals their conformational variability as a tool to increase enzyme selectivity
(
347 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366linking, 1475-6374electronic)
,
2019 Dec;
34(1): 1498-1505.
Impact Factor:
4.027
View
Export to BibTeX
Export to EndNote
Buemi MR,
Di Fiore A
,
De Luca L
, Angeli A, Mancuso F, Ferro S,
Monti SM
,
Buonanno M
, Russo E, De Sarro G,
De Simone G
, Supuran CT, Gitto R
*
Exploring structural properties of potent human carbonic anhydrase inhibitors bearing a 4-(cycloalkylamino-1-carbonyl)benzenesulfonamide moiety
(
494 views
)
Eur J Med Chem (ISSN: 1768-3254electronic, 0223-5234linking)
,
2019 Feb 1;
163: 443-452.
Impact Factor:
4.833
View
Export to BibTeX
Export to EndNote
De Simone G
*
Targeted treatment of anaerobic cancer. Patent evaluation of US2016279084 and US2017056350
(
330 views
)
Expert Opin Ther Pat (ISSN: 1744-7674electronic, 1354-3776linking)
,
2019 Jan;
29(1): 1-6.
Impact Factor:
3.699
View
Export to BibTeX
Export to EndNote
Alterio V
,
Esposito D
,
Monti SM
, Supuran CT,
De Simone G
*
Crystal structure of the human carbonic anhydrase II adduct with 1-(4-sulfamoylphenyl-ethyl)-2, 4, 6-triphenylpyridinium perchlorate, a membrane-impermeant, isoform selective inhibitor
(
638 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6374electronic, 1475-6366linking)
,
2018 Dec;
33(1): 151-157.
Impact Factor:
4.293
View
Export to BibTeX
Export to EndNote
Monti SM
, Meccariello A, Ceruso M, Szafranski K, Slawinski J, Supuran CT
*
Inhibition studies of Brucella suis beta-carbonic anhydrases with a series of 4-substituted pyridine-3-sulphonamides
(
480 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6374electronic, 1475-6366linking)
,
2018 Dec;
33(1): 255-259.
Impact Factor:
2.332
View
Export to BibTeX
Export to EndNote
Angeli A,
Buonanno M
, Donald WA,
Monti SM
, Supuran CT
*
The zinc - but not cadmium - containing zeta-carbonic from the diatom Thalassiosira weissflogii is potently activated by amines and amino acids
(
367 views
)
Bioorg Chem (ISSN: 1090-2120electronic, 0045-2068linking)
,
2018 Oct;
80: 261-265.
Impact Factor:
3.929
View
Export to BibTeX
Export to EndNote
De Simone G
, Angeli A, Bozdag M, Supuran CT, Winum JY,
Monti SM
,
Alterio V
*
Inhibition of carbonic anhydrases by a substrate analog: benzyl carbamate directly coordinates the catalytic zinc ion mimicking bicarbonate binding
(
322 views
)
Chem Commun (ISSN: 1364-548xelectronic, 1359-7345linking)
,
2018 Sep 11;
54(73): 10312-10315.
Impact Factor:
6.169
View
Export to BibTeX
Export to EndNote
Langella E
,
Buonanno M
, Vullo D, Dathan N,
Leone M
, Supuran C,
De Simone G
,
Monti SM
*
Biochemical, biophysical and molecular dynamics studies on the proteoglycan-like domain of carbonic anhydrase IX
(
413 views
)
Cell Mol Life Sci (ISSN: 1420-682xlinking)
,
2018 Sep;
75(17): 3283-3296.
Impact Factor:
6.721
View
Export to BibTeX
Export to EndNote
Supuran CT,
Alterio V
,
Di Fiore A
,
D'Ambrosio K
, Carta F,
Monti SM
,
De Simone G
*
Inhibition of carbonic anhydrase IX targets primary tumors, metastases, and cancer stem cells: Three for the price of one
(
808 views
)
Med Res Rev (ISSN: 1098-1128electronic, 0198-6325linking)
,
2018 Sep;
38(6): 1799-1836.
Impact Factor:
8.29
View
Export to BibTeX
Export to EndNote
Mishra CB, Kumari S, Angeli A, Bua S,
Buonanno M
,
Monti SM
, Tiwari M, Supuran CT
*
Discovery of potent anti-convulsant carbonic anhydrase inhibitors: Design, synthesis, in vitro and in vivo appraisal
(
380 views
)
Eur J Med Chem (ISSN: 0223-5234linking, 1768-3254electronic)
,
2018 Aug 5;
156: 430-443.
Impact Factor:
4.816
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Monti DM, Scaloni A,
De Simone G
,
Monti SM
*
Protective Role of Carbonic Anhydrases III and VII in Cellular Defense Mechanisms upon Redox Unbalance
(
298 views
)
Oxid Med Cell Longev (ISSN: 1942-0994linking)
,
2018 Aug 5;
2018:2018306: 2018306-2018306.
Impact Factor:
4.936
View
Export to BibTeX
Export to EndNote
Buonanno M
,
Di Fiore A
,
Langella E
, D’ambrosio K, Supuran CT,
Monti SM
,
De Simone G
*
The Crystal Structure of a hCA VII Variant Provides Insights into the Molecular Determinants Responsible for Its Catalytic Behavior
(
507 views
)
Int J Mol Sc (ISSN: 1661-6596, 1422-0067, 1422-0067electronic)
,
2018 May;
19(6): 19-24.
Impact Factor:
3.687
View
Export to BibTeX
Export to EndNote
Squeglia F
,
Ruggiero A
, De Simone A,
Berisio R
*
A structural overview of mycobacterial adhesins: Key biomarkers for diagnostics and therapeutics
(
344 views
)
Protein Sci (ISSN: 1469-896xelectronic, 0961-8368linking)
,
2018 Feb;
27(2): 369-380.
Impact Factor:
2.523
View
Export to BibTeX
Export to EndNote
Lanza V, Bellia F, Rizzarelli E
*
An inorganic overview of natural Aβ fragments: Copper(II) and zinc(II)-mediated pathways
(
1005 views
)
Coord Chem Rev (ISSN: 0010-8545)
,
2018;
369: 1-14.
Impact Factor:
11.225
View
Export to BibTeX
Export to EndNote
D'Ambrosio K
, Supuran CT,
De Simone G
*
Are Carbonic Anhydrases Suitable Targets to Fight Protozoan Parasitic Diseases?
(
334 views
)
Curr Med Chem (ISSN: 1875-533xelectronic, 0929-8673linking)
,
2018;
25(39): 5266-5278.
Impact Factor:
4.63
View
Export to BibTeX
Export to EndNote
De Simone G
,
Langella E
,
Esposito D
, Supuran CT,
Monti SM
, Winum JY,
Alterio V
*
Insights into the binding mode of sulphamates and sulphamides to hCA II: crystallographic studies and binding free energy calculations
(
336 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366, 1475-6374electronic, 1475-6366linking)
,
2017 Dec;
32(1): 1002-1011.
Impact Factor:
3.638
View
Export to BibTeX
Export to EndNote
Monti DM,
De Simone G
,
Langella E
, Supuran CT,
Di Fiore A
,
Monti SM
*
Insights into the role of reactive sulfhydryl groups of Carbonic Anhydrase III and VII during oxidative damage
(
482 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366, 1475-6374electronic, 1475-6366linking)
,
2017 Dec;
32(1): 5-12.
Impact Factor:
3.638
View
Export to BibTeX
Export to EndNote
Brunò E, Buemi MR,
Di Fiore A
, De LucaL, Ferro S, Angeli A, Cirilli R, Sadutto D,
Alterio V
,
Monti SM
, Supuran CT,
De Simone G
, Gitto R
*
Probing Molecular Interactions between Human Carbonic Anhydrases (hCAs) and a Novel Class of Benzenesulfonamides
(
541 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2017 May 25;
60(10): 4316-4326.
Impact Factor:
6.253
View
Export to BibTeX
Export to EndNote
Buonanno M
,
Langella E
, Zambrano N, Succoio M, Sasso E,
Alterio V
,
Di Fiore A
,
Sandomenico A
, Supuran CT, Scaloni A,
Monti SM
,
De Simone G
*
Disclosing the Interaction of Carbonic Anhydrase IX with Cullin-Associated NEDD8-Dissociated Protein 1 by Molecular Modeling and Integrated Binding Measurements
(
488 views
)
Acs Chem Biol (ISSN: 1554-8929)
,
2017 Apr 19;
N/D: N/D-N/D.
Impact Factor:
4.592
View
Export to BibTeX
Export to EndNote
Mishra CB, Kumari S, Angeli A,
Monti SM
,
Buonanno M
, Tiwari M, Supuran CT
*
Discovery of Benzenesulfonamides with Potent Human Carbonic Anhydrase Inhibitory and Effective Anticonvulsant Action: Design, Synthesis, and Pharmacological Assessment
(
1075 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2017 Mar 23;
60(6): 2456-2469.
Impact Factor:
6.253
View
Export to BibTeX
Export to EndNote
Altug C, Gunes H, Nocentini A,
Monti SM
,
Buonanno M
, Supuran CT
*
Synthesis of isoxazole-containing sulfonamides with potent carbonic anhydrase II and VII inhibitory properties
(
390 views
)
Bioorg Med Chem (ISSN: 0968-0896, 1464-3391, 0968-0896linking)
,
2017 Feb 15;
25(4): 1456-1464.
Impact Factor:
2.881
View
Export to BibTeX
Export to EndNote
Angapelly S, Ramya PV, Angeli A,
Monti SM
,
Buonanno M
, Alvala M, Supuran CT, Arifuddin M
*
Discovery of 4-sulfamoyl-phenyl-beta-lactams as a new class of potent carbonic anhydrase isoforms I, II, IV and VII inhibitors: The first example of subnanomolar CA IV inhibitors
(
400 views
)
Bioorg Med Chem (ISSN: 0968-0896, 1464-3391, 0968-0896linking)
,
2017 Jan 15;
pii:S0968-0896(16): 539-544.
Impact Factor:
2.881
View
Export to BibTeX
Export to EndNote
Angapelly S, Ramya PVS, Angeli A,
Monti SM
,
Buonanno M
, Alvala M, Supuran CT, Arifuddin M
*
Discovery of 4-sulfamoyl-phenyl-β-lactams as a new class of potent carbonic anhydrase isoforms I, II, IV and VII inhibitors: The first example of subnanomolar CA IV inhibitors
(
333 views
)
Bioorg Med Chem (ISSN: 0968-0896, 1464-3391, 0968-0896linking)
,
2017;
25(2): 539-544.
Impact Factor:
2.881
View
Export to BibTeX
Export to EndNote
Alterio V
, Cadoni R,
Esposito D
, Vullo D, Fiore AD,
Monti SM
, Caporale A,
Ruvo M
, Sechi M, Dumy P, Supuran CT,
De Simone G
, Winum JY
*
Benzoxaborole as a new chemotype for carbonic anhydrase inhibition
(
576 views
)
Chem Commun (ISSN: 1359-7345, 1364-548x, 1364-548xelectronic)
,
2016 Sep 29;
52(80): 11983-11986.
Impact Factor:
6.319
View
Export to BibTeX
Export to EndNote
Vullo D, Supuran CT, Scozzafava A,
De Simone G
,
Monti SM
,
Alterio V
, Carta F
*
Kinetic and X-ray crystallographic investigations of substituted 2-thio-6-oxo-1, 6-dihydropyrimidine-benzenesulfonamides acting as carbonic anhydrase inhibitors
(
372 views
)
Bioorg Med Chem (ISSN: 0968-0896, 1464-3391, 0968-0896linking)
,
2016 Aug 15;
24(16): 3643-3648.
Impact Factor:
2.93
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
De Simone G
,
Alterio V
, Riccio V, Winum JY, Carta F, Supuran CT
*
The anticonvulsant sulfamide JNJ-26990990 and its S, S-dioxide analog strongly inhibit carbonic anhydrases: solution and X-ray crystallographic studies
(
340 views
)
Org Biomol Chem (ISSN: 1477-0520, 1477-0539, 1477-0539electronic)
,
2016 Jun 07;
14(21): 4853-4858.
Impact Factor:
3.564
View
Export to BibTeX
Export to EndNote
Del Prete S, De Luca V,
De Simone G
, Supuran CT, Capasso C
*
Cloning, expression and purification of the complete domain of the eta-carbonic anhydrase from Plasmodium falciparum
(
589 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366, 1475-6374electronic, 1475-6366linking)
,
2016 Jun;
31(sup4): 54-59.
Impact Factor:
4.293
View
Export to BibTeX
Export to EndNote
Langella E
,
D'Ambrosio K
, D'Ascenzio M, Carradori S,
Monti SM
, Supuran CT,
De Simone G
*
A Combined Crystallographic and Theoretical Study Explains the Capability of Carboxylic Acids to Adopt Multiple Binding Modes in the Active Site of Carbonic Anhydrases
(
433 views
)
Chemistry (ISSN: 0947-6539, 1521-3765, 1521-3765electronic)
,
2016 Jan 4;
22(1): 97-100.
Impact Factor:
5.317
View
Export to BibTeX
Export to EndNote
Mishra CB, Kumari S, Angeli A,
Monti SM
,
Buonanno M
, Prakash A, Tiwari M, Supuran CT
*
Design, synthesis and biological evaluation of N-(5-methyl-isoxazol-3-yl/1, 3, 4-thiadiazol-2-yl)-4-(3-substitutedphenylureido) benzenesulfonamides as human carbonic anhydrase isoenzymes I, II, VII and XII inhibitors
(
396 views
)
J Enzyme Inhib Med Chem
,
2016;
17: 1-6.
Impact Factor:
3.428
View
Export to BibTeX
Export to EndNote
Mollica A, Locatelli M, Macedonio G, Carradori S, Sobolev AP, De Salvador RF,
Monti SM
,
Buonanno M
, Zengin G, Angeli A, Supuran CT
*
Microwave-assisted extraction, HPLC analysis, and inhibitory effects on carbonic anhydrase I, II, VA, and VII isoforms of 14 blueberry Italian cultivars
(
341 views
)
J Enzyme Inhib Med Chem
,
2016;
31(sup4): N/D-N/D.
Impact Factor:
3.428
View
Export to BibTeX
Export to EndNote
La Regina G, Coluccia A, Famiglini V, Pelliccia S, Monti L, Vullo D, Nuti E,
Alterio V
,
De Simone G
,
Monti SM
, Pan P, Parkkila S, Supuran CT, Rossello A, Silvestri R
*
Discovery of 1, 1'-Biphenyl-4-sulfonamides as a New Class of Potent and Selective Carbonic Anhydrase XIV Inhibitors
(
428 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2015 Nov 12;
58(21): 8564-8572.
Impact Factor:
5.589
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
Vergara A
, Caterino M,
Alterio V
,
Monti SM
, Ombouma J, Dumy P, Vullo D, Supuran CT, Winum JY,
De Simone G
*
Hydroxylamine-O-sulfonamide is a versatile lead compound for the development of carbonic anhydrase inhibitors
(
434 views
)
(PDF
254 views
)
Chem Commun (ISSN: 1359-7345, 1364-548x, 1364-548xelectronic)
,
2015 Jul 2;
51(57): 11519-11522.
Impact Factor:
6.567
View
Export to BibTeX
Export to EndNote
De Simone G
,
Monti SM
,
Alterio V
,
Buonanno M
, De Luca V, Rossi M, Carginale V, Supuran CT, Capasso C,
Di Fiore A
*
Crystal structure of the most catalytically effective carbonic anhydrase enzyme known, SazCA from the thermophilic bacterium Sulfurihydrogenibium azorense
(
420 views
)
Bioorg Med Chem Lett (ISSN: 0960-894x)
,
2015 May 1;
25(9): 2002-2006.
Impact Factor:
2.486
View
Export to BibTeX
Export to EndNote
Alterio V
, Tanc M, Ivanova J, Zalubovskis R, Vozny I,
Monti SM
,
Di Fiore A
,
De Simone G
, Supuran CT
*
X-ray crystallographic and kinetic investigations of 6-sulfamoyl-saccharin as a carbonic anhydrase inhibitor
(
485 views
)
Org Biomol Chem (ISSN: 1477-0520, 1477-0539, 1477-0539electronic)
,
2015 Apr 7;
13(13): 4064-4069.
Impact Factor:
3.559
View
Export to BibTeX
Export to EndNote
De Simone G
,
Di Fiore A
, Capasso C, Supuran CT
*
The zinc coordination pattern in the eta-carbonic anhydrase from Plasmodium falciparum is different from all other carbonic anhydrase genetic families
(
589 views
)
Bioorg Med Chem Lett (ISSN: 0960-894x)
,
2015 Apr 1;
25(7): 1385-1389.
Impact Factor:
2.486
View
Export to BibTeX
Export to EndNote
Alterio V
,
Langella E
,
De Simone G
,
Monti SM
*
Cadmium-containing carbonic anhydrase CDCA1 in marine diatom Thalassiosira weissflogii
(
876 views
)
Mar Drugs (ISSN: 1660-3397, 1660-3397linking)
,
2015 Mar 25;
13(4): 1688-1697.
Impact Factor:
3.345
View
Export to BibTeX
Export to EndNote
Monti SM
, Supuran CT, De Simone G
*
DPP-4 inhibitors: a patent review (2012 - 2014)
(
649 views
)
Expert Opin Ther Pat (ISSN: 1354-3776, 1744-7674electronic)
,
2015 Feb;
25(2): 209-236.
Impact Factor:
4.626
View
Export to BibTeX
Export to EndNote
Supuran CT, Capasso C,
De Simone G
*
Carbonic Anhydrase II as Target for Drug Design
(
403 views
)
Carbonic Anhydrases As Biocatalysts
,
2015 Jan 08;
N/D: 51-90.
Impact Factor:
0
View
Export to BibTeX
Export to EndNote
Monti SM
, Supuran CT,
De Simone G
,
Di Fiore A
*
Carbonic Anhydrase VII
(
306 views
)
Carbonic Anhydrases As Biocatalysts
,
2015 Jan 08;
N/D: 151-168.
Impact Factor:
0
View
Export to BibTeX
Export to EndNote
D'Ambrosio K
,
De Simone G
, Supuran CT
*
Human Carbonic Anhydrases: Catalytic Properties, Structural Features, and Tissue Distribution
(
438 views
)
Carbonic Anhydrases As Biocatalysts
,
2015 Jan 08;
N/D: 17-30.
Impact Factor:
0
View
Export to BibTeX
Export to EndNote
D'Ambrosio K
, Carradori S,
Monti SM
,
Buonanno M
, Secci D, Vullo D, Supuran CT,
De Simone G
*
Out of the active site binding pocket for carbonic anhydrase inhibitors
(
674 views
)
(PDF
264 views
)
Chem Commun (ISSN: 1359-7345, 1364-548x, 1364-548xelectronic)
,
2015 Jan 7;
51(2): 302-305.
Impact Factor:
6.567
View
Export to BibTeX
Export to EndNote
Ceruso M, Carta F, Osman SM, Alothman Z,
Monti SM
, Supuran CT
*
Inhibition studies of bacterial, fungal and protozoan β-class carbonic anhydrases with Schiff bases incorporating sulfonamide moieties
(
498 views
)
Bioorg Med Chem (ISSN: 0968-0896, 1464-3391, 0968-0896linking)
,
2015;
23(15): 4181-4187.
Impact Factor:
2.923
View
Export to BibTeX
Export to EndNote
Iqbal J, Al-rashida M, Durdagi S,
Alterio V
,
Di Fiore A
*
Recent developments of carbonic anhydrase inhibitors as potential drugs
(
704 views
)
Biomed Res Int (ISSN: 2314-6133, 2314-6141)
,
2015;
2015: 174178-174178.
Impact Factor:
2.134
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
Alterio V
,
Monti SM
,
De Simone G
, D’Ambrosio K
*
Thermostable carbonic anhydrases in biotechnological applications
(
636 views
)
Int J Mol Sc (ISSN: 1422-0067, 1661-6596, 1422-0067linking)
,
2015;
16(7): 15456-15480.
Impact Factor:
3.257
View
Export to BibTeX
Export to EndNote
Musumeci D
,
Roviello GN
, Montesarchio D
*
An overview on HMGB1 inhibitors as potential therapeutic agents in HMGB1-related pathologies
(
655 views
)
Pharmacol Ther (ISSN: 0163-7258, 0163-7258linking)
,
2014 Mar;
141(3): 347-357.
Impact Factor:
9.723
View
Export to BibTeX
Export to EndNote
Dathan NA,
Alterio V
, Troiano E, Vullo D, Ludwig M,
De Simone G
, Supuran CT,
Monti SM
*
Biochemical Characterization Of The Chloroplastic β-Carbonic Anhydrase From Flaveria Bidentis (l. ) "kuntze"
(
693 views
)
J Enzym Inhib Med Ch (ISSN: 1475-6366, 1475-6374electronic, 1475-6366linking)
,
2014;
29(4): 500-504.
Impact Factor:
2.332
View
Export to BibTeX
Export to EndNote
De Simone G
, Pizika G,
Monti SM
,
Di Fiore A
, Ivanova J, Vozny I, Trapencieris P, Zalubovskis R, Supuran CT,
Alterio V
*
Hydrophobic substituents of the phenylmethylsulfamide moiety can be used for the development of new selective carbonic anhydrase inhibitors
(
419 views
)
Biomed Res Int (ISSN: 2314-6133, 2314-6141)
,
2014;
2014: 523210-523210.
Impact Factor:
1.579
View
Export to BibTeX
Export to EndNote
Alterio V
, Pan P, Parkkila S,
Buonanno M
, Supuran CT,
Monti SM
,
De Simone G
*
The Structural Comparison Between Membrane-Associated Human Carbonic Anhydrases Provides Insights Into Drug Design Of Selective Inhibitors
(
562 views
)
Biopolymers (ISSN: 0006-3525, 0006-6352, 0006-3525print)
,
2014;
101(7): 769-778.
Impact Factor:
2.385
View
Export to BibTeX
Export to EndNote
Alterio V
,
Monti SM
,
De Simone G
*
Thermal-stable carbonic anhydrases: a structural overview
(
468 views
)
Subcell Biochem (ISSN: 0306-0225)
,
2014;
75: 387-404.
Impact Factor:
33.116
View
Export to BibTeX
Export to EndNote
Rami M, Dubois L, Parvathaneni NK,
Alterio V
, van Kuijk SJ,
Monti SM
, Lambin P,
De Simone G
, Supuran CT, Winum JY
*
Hypoxia-targeting carbonic anhydrase IX inhibitors by a new series of nitroimidazole-sulfonamides/sulfamides/sulfamates
(
668 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2013 Nov 14;
56(21): 8512-8520.
Impact Factor:
5.48
View
Export to BibTeX
Export to EndNote
De Simone G
,
Alterio V
, Supuran CT
*
Exploiting the hydrophobic and hydrophilic binding sites for designing carbonic anhydrase inhibitors
(
650 views
)
Expert Opin Drug Discov (ISSN: 1746-0441)
,
2013 Jul;
8(7): 793-810.
Impact Factor:
3.467
View
Export to BibTeX
Export to EndNote
Monti SM
, Supuran CT,
De Simone G
*
Anticancer carbonic anhydrase inhibitors: A patent review (2008-2013)
(
607 views
)
Expert Opin Ther Pat (ISSN: 1354-3776, 1744-7674electronic)
,
2013 Jun;
23(6): 737-749.
Impact Factor:
3.441
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Capasso C, De Luca V,
Monti SM
, Carginale V, Supuran CT, Scozzafava A,
Pedone C
, Rossi M,
De Simone G
*
X-ray structure of the first 'extremo-alpha-carbonic anhydrase', a dimeric enzyme from the thermophilic bacterium Sulfurihydrogenibium yellowstonense YO3AOP1
(
904 views
)
Acta Crystallogr D Biol Crystallogr (ISSN: 0907-4449, 0907-4449linking)
,
2013 Jun;
69(6): 1150-1159.
Impact Factor:
7.232
View
Export to BibTeX
Export to EndNote
Russo Krauss I
,
Merlino A
,
Vergara A
,
Sica F
*
An overview of biological macromolecule crystallization
(
1352 views
)
Int J Mol Sc (ISSN: 1422-0067, 1661-6596, 1422-0067electronic)
,
2013 May 31;
14(6): 11643-11691.
Impact Factor:
2.339
View
Export to BibTeX
Export to EndNote
Monti SM
,
De Simone G
, Dathan NA, Ludwig M, Vullo D, Scozzafava A, Capasso C, Supuran CT
*
Kinetic And Anion Inhibition Studies Of A Beta-Carbonic Anhydrase (fbica 1) From The C-4 Plant Flaveria Bidentis
(
553 views
)
Bioorg Med Chem Lett (ISSN: 0960-894x)
,
2013 Mar 15;
23(6): 1626-1630.
Impact Factor:
2.331
View
Export to BibTeX
Export to EndNote
Bartolucci S, Contursi P, Fiorentino G, Limauro D,
Pedone E
*
Responding to toxic compounds: a genomic and functional overview of Archaea
(
884 views
)
Frontiers In Bioscience (ISSN: 1093-9946, 1093-4715)
,
2013 Jan 1;
18: 165-189.
Impact Factor:
4.249
View
Export to BibTeX
Export to EndNote
Buanne P, Renzone G, Monteleone F, Vitale M,
Monti SM
,
Sandomenico A
, Garbi C, Montanaro D, Accardo M, Troncone G, Zatovicova M, Csaderova L, Supuran CT, Pastorekova S, Scaloni A,
De Simone G
, Zambrano N
*
Characterization of carbonic anhydrase ix interactome reveals proteins assisting its nuclear localization in hypoxic cells
(
590 views
)
J Proteome Res (ISSN: 1535-3893)
,
2013 Jan;
12(1): 282-292.
Impact Factor:
5.001
View
Export to BibTeX
Export to EndNote
Del Giudice R, Monti DM, Truppo E, Arciello A, Supuran CT,
De Simone G
,
Monti SM
*
Human Carbonic Anhydrase Vii Protects Cells From Oxidative Damage
(
451 views
)
Biol Chem Biological Chemistry (ISSN: 1431-6730, 1431-1673, 1437-4315)
,
2013;
394(10): 1343-1348.
Impact Factor:
2.689
View
Export to BibTeX
Export to EndNote
Alterio V
,
Di Fiore A
,
D'Ambrosio K
, Supuran CT,
De Simone G
*
Multiple binding modes of inhibitors to carbonic anhydrases: How to design specific drugs targeting 15 different isoforms?
(
666 views
)
Chem Rev (ISSN: 0009-2665)
,
2012 Sep;
112(8): 4421-4468.
Impact Factor:
41.298
View
Export to BibTeX
Export to EndNote
Ruggiero A
, Smaldone G,
Squeglia F
,
Berisio R
*
Enhanced crystallizability by protein engineering approaches: A general overview
(
2195 views
)
Protein Pept Lett (ISSN: 0929-8665, 1875-5305)
,
2012 Jul;
19(7): 732-742.
Impact Factor:
1.994
View
Export to BibTeX
Export to EndNote
De Simone G
, Supuran CT
*
(In)organic anions as carbonic anhydrase inhibitors
(
548 views
)
J Chem Res (ISSN: 0162-0134, 1873-3344, 0162-0134print)
,
2012 Jun;
111: 117-129.
Impact Factor:
3.197
View
Export to BibTeX
Export to EndNote
Alterio V
,
Langella E
, Viparelli F, Vullo D, Ascione G, Dathan NA, Morel FM, Supuran CT,
De Simone G
,
Monti SM
*
Structural and inhibition insights into carbonic anhydrase CDCA1 from the marine diatom Thalassiosira weissflogii
(
635 views
)
Biochimie (ISSN: 0300-9084, 1638-6183, 1638-6183electronic)
,
2012 May;
94(5): 1232-1241.
Impact Factor:
3.142
View
Export to BibTeX
Export to EndNote
Truppo E, Supuran CT,
Sandomenico A
, Vullo D, Innocenti A,
Di Fiore A
,
Alterio V
,
De Simone G
,
Monti SM
*
Carbonic anhydrase VII is S-glutathionylated without loss of catalytic activity and affinity for sulfonamide inhibitors
(
497 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2012 Feb 15;
22(4): 1560-1564.
Impact Factor:
2.338
View
Export to BibTeX
Export to EndNote
Monti SM
, Supuran CT,
De Simone G
*
Carbonic anhydrase IX as a target for designing novel anticancer drugs
(
885 views
)
Curr Med Chem (ISSN: 0929-8673, 1875-533x, 1875-533xelectronic)
,
2012 Feb;
19(6): 821-830.
Impact Factor:
4.07
View
Export to BibTeX
Export to EndNote
De Simone G
*
Editorial: Zinc Metallo-Enzymes As Target For Drug Design
(
578 views
)
Curr Med Chem (ISSN: 0929-8673, 1875-533x, 1875-533xelectronic)
,
2012 Feb;
19(6): 820-1012.
Impact Factor:
4.07
View
Export to BibTeX
Export to EndNote
Monti SM
, Maresca A, Viparelli F, Carta F,
De Simone G
, Muehlschlegel FA, Scozzafava A, Supuran CT
*
Dithiocarbamates are strong inhibitors of the beta-class fungal carbonic anhydrases from Cryptococcus neoformans, Candida albicans and Candida glabrata
(
511 views
)
Bioorg Med Chem Lett (ISSN: 0960-894x)
,
2012 Jan 15;
22(2): 859-862.
Impact Factor:
2.338
View
Export to BibTeX
Export to EndNote
D'Ambrosio K
, Smaine F-Z, Carta F,
De Simone G
, Winum J-Y, Supuran CT
*
Development of potent carbonic anhydrase inhibitors incorporating both sulfonamide and sulfamide groups
(
574 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2012;
55(15): 6776-6783.
Impact Factor:
5.614
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Maresca A, Supuran CT,
De Simone G
*
Hydroxamate represents a versatile zinc binding group for the development of new carbonic anhydrase inhibitors
(
438 views
)
Chem Commun (ISSN: 1359-7345, 1364-548x, 1364-548xelectronic)
,
2012;
48(70): 8838-8840.
Impact Factor:
6.378
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Maresca A,
Alterio V
, Supuran CT,
De Simone G
*
Carbonic anhydrase inhibitors: X-ray crystallographic studies for the binding of N-substituted benzenesulfonamides to human isoform II
(
406 views
)
Chem Commun (ISSN: 1359-7345, 1364-548x, 1364-548xelectronic)
,
2011;
47(42): 11636-11638.
Impact Factor:
6.169
View
Export to BibTeX
Export to EndNote
Viparelli F,
Monti SM
,
De Simone G
, Innocenti A, Scozzafava A, Xu Y, Morel FMM, Supuran CT
*
Inhibition Of The R1 Fragment Of The Cadmium-Containing Zeta-Class Carbonic Anhydrase From The Diatom Thalassiosira Weissflogii With Anions
(
399 views
)
Bioorganic & Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2010 Sep 15;
20(16): 4745-4748.
Impact Factor:
2.661
View
Export to BibTeX
Export to EndNote
Alterio V
,
Monti SM
, Truppo E,
Pedone C
, Supuran CT,
De Simone G
*
The first example of a significant active site conformational rearrangement in a carbonic anhydrase-inhibitor adduct: The carbonic anhydrase I-topiramate complex
(
638 views
)
Org Biomol Chem (ISSN: 1477-0520, 1477-0539, 1477-0539electronic)
,
2010 Sep 7;
8(15): 3528-3533.
Impact Factor:
3.451
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Truppo E, Supuran CT,
Alterio V
, Dathan N, Bootorabi F, Parkkila S,
Monti SM
,
De Simone G
*
Crystal structure of the C183S/C217S mutant of human CA VII in complex with acetazolamide
(
565 views
)
Bioorg Med Chem Lett (ISSN: 0960-894x)
,
2010 Sep 1;
20(17): 5023-5026.
Impact Factor:
2.661
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
Monti SM
, Innocenti A, Winum J-Y,
De Simone G
, Supuran CT
*
Carbonic anhydrase inhibitors: Crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV
(
428 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2010 Jun 15;
20(12): 3601-3605.
Impact Factor:
2.661
View
Export to BibTeX
Export to EndNote
Roviello GN
, Benedetti E,
Pedone C
, Bucci EM
*
Nucleobase-containing peptides: An overview of their characteristic features and applications
(
1047 views
)
Amino Acids (ISSN: 0939-4451, 1438-2199, 1438-2199electronic)
,
2010 Jun;
39(1): 45-57.
Impact Factor:
4.106
View
Export to BibTeX
Export to EndNote
De Simone G
, Supuran CT
*
Carbonic anhydrase IX: Biochemical and crystallographic characterization of a novel antitumor target
(
534 views
)
Bba-Gen Subjects (ISSN: 1570-9639, 0006-3002, 0925-4439)
,
2010 Feb;
1804(2): 404-409.
Impact Factor:
2.773
View
Export to BibTeX
Export to EndNote
Guler OO,
De Simone G
, Supuran CT
*
Drug design studies of the novel antitumor targets carbonic anhydrase IX and XII
(
636 views
)
Curr Med Chem (ISSN: 0929-8673, 1875-533x, 1875-533xelectronic)
,
2010;
17(15): 1516-1526.
Impact Factor:
4.63
View
Export to BibTeX
Export to EndNote
Supuran CT,
Di Fiore A
,
Alterio V
,
Monti SM
,
De Simone G
*
Recent advances in structural studies of the carbonic anhydrase family: The crystal structure of human CA IX and CA XIII
(
609 views
)
Curr Pharm Des Current Pharmaceutical Design (ISSN: 1381-6128, 1873-4286)
,
2010;
16(29): 3246-3254.
Impact Factor:
4.774
View
Export to BibTeX
Export to EndNote
Innocenti A, Pastorekova S, Pastorek J, Scozzafava A,
De Simone G
, Supuran CT
*
The proteoglycan region of the tumor-associated carbonic anhydrase isoform IX acts as anintrinsic buffer optimizing CO2 hydration at acidic pH values characteristic of solid tumors
(
383 views
)
Bioorganic & Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2009 Oct 15;
19(20): 5825-5828.
Impact Factor:
2.65
View
Export to BibTeX
Export to EndNote
Vitale RM,
Alterio V
, Innocenti A, Winum JY,
Monti SM
,
De Simone G
, Supuran CT
*
Carbonic anhydrase inhibitors. Comparison of aliphatic sulfamate/bis- sulfamate adducts with isozymes II and IX as a platform for designing tight-binding, more isoform-selective inhibitors
(
563 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2009 Oct 8;
52(19): 5990-5998.
Impact Factor:
4.802
View
Export to BibTeX
Export to EndNote
Alterio V
, Hilvo M,
Di Fiore A
, Supuran CT, Pan P, Parkkila S, Scaloni A, Pastorek J, Pastorekova S,
Pedone C
, Scozzafava A,
Monti SM
,
De Simone G
*
Crystal structure of the catalytic domain of the tumor-associated human carbonic anhydrase IX
(
723 views
)
P Natl Acad Sci Usa (ISSN: 0027-8424, 1091-6490, 0027-8424print)
,
2009 Sep 22;
106(38): 16233-16238.
Impact Factor:
9.432
View
Export to BibTeX
Export to EndNote
De Simone G
, Scozzafava A, Supuran CT
*
Which Carbonic Anhydrases are Targeted by the Antiepileptic Sulfonamides and Sulfamates?
(
506 views
)
Chem Biol Drug Des (ISSN: 1747-0277, 1747-0285)
,
2009 Sep;
74(3): 317-321.
Impact Factor:
2.473
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
Monti SM
, Hilvo M, Parkkila S, Romano V, Scaloni A,
Pedone C
, Scozzafava A, Supuran CT,
De Simone G
*
Crystal structure of human carbonic anhydrase XIII and its complex with the inhibitor acetazolamide
(
987 views
)
Proteins (ISSN: 1097-0134, 0887-3585, 1097-0134electronic)
,
2009 Jan;
74(1): 164-175.
Impact Factor:
3.085
View
Export to BibTeX
Export to EndNote
Hilvo M,
De Simone G
, Supuran CT, Parkkila S
*
Advances in the Inhibitory and Structural Investigations on Carbonic Anhydrase Isozymes XIII and XV
(
380 views
)
Drug Des Of Zinc Enzyme Inhibitors (ISSN: 9780-4702, 9780-470275009)
,
2009;
N/D: 273-283.
Impact Factor:
1.156
View
Export to BibTeX
Export to EndNote
De Simone G
, Supuran CT
*
Drug Design of Antiobesity Carbonic Anhydrase Inhibitors
(
429 views
)
Drug Des Of Zinc Enzyme Inhibitors (ISSN: 9780-4702, 9780-470275009)
,
2009;
66(DECEMBERSPEC.I): 241-254.
Impact Factor:
1.156
View
Export to BibTeX
Export to EndNote
Alterio V
,
Di Fiore A
,
D'Ambrosio K
, Supuran CT,
De Simone G
*
X-Ray Crystallography of Carbonic Anhydrase Inhibitors and Its Importance in Drug Design
(
529 views
)
Drug Des Of Zinc Enzyme Inhibitors (ISSN: 9780-4702, 9780-470275009)
,
2009;
N/D: 73-138.
Impact Factor:
1.156
View
Export to BibTeX
Export to EndNote
Hilvo M, Baranauskiene L, Salzano AM, Scaloni A, Matulis D, Innocenti A, Scozzafava A,
Monti SM
,
Di Fiore A
,
De Simone G
, Lindfors M, Janis J, Valjakka J, Pastorekova S, Pastorek J, Kulomaa MS, Nordlund HR, Supuran CT, Parkkila S
*
Biochemical characterization of CA IX, one of the most active carbonic anhydrase isozymes
(
896 views
)
Jbc Papers (ISSN: 0021-9258, 1083-351x, 0021-9258linking)
,
2008 Oct 10;
283(41): 27799-27809.
Impact Factor:
5.52
View
Export to BibTeX
Export to EndNote
D'Ambrosio K
, Vitale R, Dogne J, Masereel B, Innocenti A, Scozzafava A,
De Simone G
, Supuran CT
*
Ccarbonic Anhydrase Inhibitors: Bioreductive Nitro-Containing Sulfonamides With Selectivity For Targeting The Tumor Associated Isoforms Ix And Xii
(
1009 views
)
J Med Chem (ISSN: 1520-4804, 0022-2623, 0022-2623print)
,
2008 Jun 12;
51(11): 3230-3237.
Impact Factor:
4.898
View
Export to BibTeX
Export to EndNote
Supuran CT,
Di Fiore A
,
De Simone G
*
Carbonic anhydrase inhibitors as emerging drugs for the treatment of obesity
(
762 views
)
Expert Opin Emerg Drugsexpert Opinion On Emerging Drugs (ISSN: 1472-8214)
,
2008 Jun;
13(2): 383-392.
Impact Factor:
3.08
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
Pedone C
, Antel J, Waldeck H, Witte A, Wurl M, Scozzafava A, Supuran CT,
De Simone G
*
Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors
(
535 views
)
Bioorg Med Chem Lett (ISSN: 1464-3405, 0960-894x, 1464-3405electronic)
,
2008 Apr 15;
18(8): 2669-2674.
Impact Factor:
2.531
View
Export to BibTeX
Export to EndNote
Innocenti A, Scozzafava A, Parkkila S, Puccetti L,
De Simone G
, Supuran CT
*
Investigations of the esterase, phosphatase, and sulfatase activities of the cytosolic mammalian carbonic anhydrase isoforms I, II, and XIII with 4-nitrophenyl esters as substrates
(
491 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2008 Apr 1;
18(7): 2267-2271.
Impact Factor:
2.531
View
Export to BibTeX
Export to EndNote
Leese MP, Jourdan FL, Gaukroger K, Mahon MF, Newman SP, Foster PA, Stengel C, Regis-Lydi S, Ferrandis E,
Di Fiore A
,
De Simone G
, Supuran CT, Purohit A, Reed MJ, Potter BVL
*
Structure-activity relationships of C-17 cyano-substituted estratrienes as anticancer agents
(
607 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2008 Mar 13;
51(5): 1295-1308.
Impact Factor:
4.898
View
Export to BibTeX
Export to EndNote
De Simone G
,
Di Fiore A
, Supuran CT
*
Are carbonic anhydrase inhibitors suitable for obtaining antiobesity drugs?
(
608 views
)
Curr Pharm Des Current Pharmaceutical Design (ISSN: 1381-6128, 1873-4286)
,
2008 Mar;
14(7): 655-660.
Impact Factor:
4.399
View
Export to BibTeX
Export to EndNote
D'Ambrosio K
, Masereel B, Thiry A, Scozzafava A, Supuran CT,
De Simone G
*
Carbonic anhydrase inhibitors: Binding of indanesulfonamides to the human isoform II
(
510 views
)
Chemmedchem (ISSN: 1860-7179, 1860-7187, 1860-7187electronic)
,
2008 Mar;
3(3): 473-477.
Impact Factor:
3.15
View
Export to BibTeX
Export to EndNote
Supuran CT,
De Simone G
Carbonic anhydrases--an overview
(
470 views
)
Curr Pharm Des
,
2008;
14(7): 603-614.
Impact Factor:
0
View
Export to BibTeX
Export to EndNote
Hilvo M, Innocenti A,
Monti SM
,
De Simone G
, Supuran CT, Parkkila S
*
Recent advances in research on the most novel carbonic anhydrases, CA XIII and XV
(
799 views
)
Curr Pharm Des Current Pharmaceutical Design (ISSN: 1381-6128, 1873-4286)
,
2008;
14(7): 672-678.
Impact Factor:
4.399
View
Export to BibTeX
Export to EndNote
Alterio V
,
De Simone G
,
Monti SM
, Scozzafava A, Supuran CT
*
Carbonic anhydrase inhibitors: Inhibition of human, bacterial, and archaeal isozymes with benzene-1, 3-disulfonamides-Solution and crystallographic studies
(
456 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2007 Sep 1;
17(15): 4201-4207.
Impact Factor:
2.604
View
Export to BibTeX
Export to EndNote
Vitale RM,
Pedone C
, Amodeo P, Antel J, Wurl M, Scozzafava A, Supuran CT,
De Simone G
*
Molecular modeling study for the binding of zonisamide and topiramate to the human mitochondrial carbonic anhydrase isoform VA
(
425 views
)
Bioorg Med Chem (ISSN: 0968-0896, 1464-3391, 1464-3391electronic)
,
2007 Jun 15;
15(12): 4152-4158.
Impact Factor:
2.662
View
Export to BibTeX
Export to EndNote
Di Fiore A
, Scozzafava A, Winum JY, Montero JL,
Pedone C
, Supuran CT,
De Simone G
*
Carbonic anhydrase inhibitors: binding of an antiglaucoma glycosyl-sulfanilamide derivative to human isoform II and its consequences for the drug design of enzyme inhibitors incorporating sugar moieties
(
536 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2007 Mar 15;
17(6): 1726-1731.
Impact Factor:
2.604
View
Export to BibTeX
Export to EndNote
De Simone G
, Supuran CT
*
Antiobesity carbonic anhydrase inhibitors
(
717 views
)
Curr Top Med Chem (ISSN: 1568-0266, 1568-0266linking, 1873-4294electronic)
,
2007;
7(9): 879-884.
Impact Factor:
4.325
View
Export to BibTeX
Export to EndNote
Leese MP, Leblond B, Smith A, Newman SP,
Di Fiore A
,
De Simone G
, Supuran CT, Purohit A, Reed MJ, Potter BVL
*
2-substituted estradiol bis-sulfamates, multitargeted antitumor agents: synthesis, in vitro SAR, protein crystallography, and in vivo activity
(
1102 views
)
J Med Chem (ISSN: 0022-2623print, 0022-2623linking, 1520-4804)
,
2006 Dec 28;
49(26): 7683-7696.
Impact Factor:
5.115
View
Export to BibTeX
Export to EndNote
Menchise V
,
De Simone G
,
Di Fiore A
, Scozzafava A, Supuran CT
*
Carbonic anhydrase inhibitors: X-ray crystallographic studies for the binding of 5-amino-1, 3, 4-thiadiazole-2-sulfonamide and 5-(4-amino-3-chloro-5-fluorophenylsulfonamido)1, 3, 4-thiadiazole-2-sulfon amide to human isoform II
(
393 views
)
Bioorganic & Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2006 Dec 15;
16(24): 6204-6208.
Impact Factor:
2.538
View
Export to BibTeX
Export to EndNote
De Simone G
, Vitale RM,
Di Fiore A
,
Pedone C
, Scozzafava A, Montero JL, Winum JY, Supuran CT
*
Carbonic anhydrase inhibitors: Hypoxia-activatable sulfonamides incorporating disulfide bonds that target the tumor-associated isoform IX
(
651 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2006 Sep 7;
49(18): 5544-5551.
Impact Factor:
5.115
View
Export to BibTeX
Export to EndNote
Alterio V
, Vitale RM,
Monti SM
,
Pedone C
, Scozzafava A, Cecchi A,
De Simone G
, Supuran CT
*
Carbonic anhydrase inhibitors: X-ray and molecular modeling study for the interaction of a fluorescent antitumor sulfonamide with isozyme II and IX
(
867 views
)
J Am Chem Soc (ISSN: 0002-7863, 0002-2786, 1520-5126)
,
2006 Jun 28;
128(25): 8329-8335.
Impact Factor:
7.696
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
Pedone C
,
D'Ambrosio K
, Scozzafava A,
De Simone G
, Supuran CT
*
Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II 'selective' inhibitor celecoxib
(
418 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2006 Jan 15;
16(2): 437-442.
Impact Factor:
2.538
View
Export to BibTeX
Export to EndNote
Menchise V
,
De Simone G
,
Alterio V
,
Di Fiore A
,
Pedone C
, Scozzafava A, Supuran CT
*
Carbonic anhydrase inhibitors: Stacking with Phe131 determines active site binding region of inhibitors as exemplified by the X-ray crystal structure of a membrane-impermeant antitumor sulfonamide complexed with isozyme II
(
600 views
)
J Med Chem (ISSN: 0022-2623, 1520-4804, 0022-2623print)
,
2005 Sep 8;
48(18): 5721-5727.
Impact Factor:
4.926
View
Export to BibTeX
Export to EndNote
De Simone G
,
Di Fiore A
,
Menchise V
,
Pedone C
, Antel J, Casini A, Scozzafava A, Wurl M, Supuran CT
*
Carbonic anhydrase inhibitors. Zonisamide is an effective inhibitor of the cytosolic isozyme II and mitochondrial isozyme V: solution and X-ray crystallographic studies
(
932 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2005 May 2;
15(9): 2315-2320.
Impact Factor:
2.478
View
Export to BibTeX
Export to EndNote
Di Fiore A
,
De Simone G
,
Menchise V
,
Pedone C
, Casini A, Scozzafava A, Supuran CT
*
Carbonic anhydrase inhibitors: X-ray crystal structure of a benzenesulfonamide strong CA II and CA IX inhibitor bearing a pentafluorophenylaminothioureido tail in complex with isozyme II
(
597 views
)
Bioorg Med Chem Lett Bioorganic And Medicinal Chemistry Letters (ISSN: 0960-894x)
,
2005 Apr 1;
15(7): 1937-1942.
Impact Factor:
2.478
View
Export to BibTeX
Export to EndNote
Acampa W
, Di Benedetto C,
Cuocolo A
An overview of radiotracers in nuclear cardiology
(
490 views
)
J Nucl Cardiol (ISSN: 1071-3581, 1532-6551, 1532-6551electronic)
,
2000 Nov;
7(6): 701-707.
Impact Factor:
1.854
View
Export to BibTeX
Export to EndNote
Fonti R
, Latella G, Caprilli R, Frieri G, Marcheggiano A, Sambuy Y
Carbonic anhydrase I reduction in colonic mucosa of patients with active ulcerative colitis
(
656 views
)
Digestive Diseases And Sciences (ISSN: 0163-2116)
,
1998;
43(9): 2086-2092.
Impact Factor:
1.972
View
Export to BibTeX
Export to EndNote
Brunetti A
,
Alfano B
, Soricelli A,
Tedeschi E
, Mainolfi C, Covelli EM, Aloj L,
Panico M
, Bazzicalupo L,
Salvatore M
Functional characterization of brain tumors: An overview of the potential clinical value
(
1018 views
)
(PDF
274 views
)
Nucl Med Biol (ISSN: 0969-8051, 0883-2897)
,
1996 Sep;
23(6): 699-715.
Impact Factor:
1.042
View
Export to BibTeX
Export to EndNote
Brunetti A
, Soricelli A, Rotondo A,
Alfano B
, Raman R, Celentano L, Di Chiro G,
Salvatore M
Correlative morphologic and functional imaging for diagnosis, staging and follow up in AIDS: an overview
(
327 views
)
Q J Nucl Med (ISSN: 1125-0135, 0392-2020, 1124-3937)
,
1995 Sep;
39(3): 201-211.
Impact Factor:
2.125
View
Export to BibTeX
Export to EndNote
140
Records (
139
excluding Abstracts).
Total impact factor:
621.682
(
616.567
excluding Abstracts).
Total 5 year impact factor:
553.399
(
547.895
excluding Abstracts).
Top of page
Copy&Paste Friendly
Export all to BibTeX
Export all to EndNote
Last modified by
Giuseppina De Simone
on Sunday 12 July 2020, 13:14:49
395 views.
Last view on Sunday 01 December 2024, 2:26:50