Synthesis, chemical characterization and biological activity of new histone acetylation/deacetylation specific inhibitors: A novel and potential approach to cancer therapy
Synthesis, chemical characterization and biological activity of new histone acetylation/deacetylation specific inhibitors: A novel and potential approach to cancer therapy(440 views) Pellerito O, Prinzivalli C, Foresti E, Sabatino P, Abbate M, Casella G, Fiore T, Scopelliti M, Pellerito C, Giuliano M, Grasso G, Pellerito L
Keywords: Esi-Ms, Mössbauer Spectroscopy, Nmr, Organotin(iv), X-Ray Spectroscopy, Antineoplastic Agent, Ester, Histone Deacetylase Inhibitor, Ligand, Lysine 14, Lysine Derivative, Organotin Compound, Tributyltin, Unclassified Drug, Valproate Ligand, Valproic Acid Derivative, Apoptosis, Article, Biological Activity, Cancer Cell Culture, Cancer Therapy, Cell Viability, Controlled Study, Crystallography, Cytotoxicity, Drug Synthesis, Histone Acetylation, Human, Human Cell, Liver Cell, Nuclear Magnetic Resonance, Solid State, Cell Survival, Hep G2 Cells, Tetra, M Ssbauer Spectroscopy, Organotin (iv),
Affiliations: *** IBB - CNR ***
Dipartimento di Biomedicina Sperimentale e Neuroscienze Cliniche, Sezione di Scienze Biochimiche, Policlinico Universitario, Via del Vespro, 129-90127 Palermo, Italy
Dipartimento di Chimica Stanislao Cannizzaro, Università Degli Studi di Palermo, Viale delle Scienze, Ed. 17, 90128 Palermo, Italy
Dipartimento di Fisica e Chimica (DiFC), Università Degli Studi di Palermo, Viale delle Scienze, Ed. 17, 90128 Palermo, Italy
Dipartimento di Scienze della Terra e Del Mare (DiSTeM), Università Degli Studi di Palermo, Viale delle Scienze, Ed. 17, 90128 Palermo, Italy
Consorzio Interuniversitario di Ricerca in Chimica Dei Metalli Nei Sistemi Biologici, Piazza Umberto I, 1-70121 Bari, Italy
Istituto di Biostrutture e Bioimmagini, CNR (C/o Dipartimento di Scienze Chimiche), Università Degli Studi di Catania, Viale Andrea Doria, 6, 95125 Catania, Italy
Department of Molecular Biology, Medical Biochemistry and Pathology, Faculty of Medicine, Université Laval, 2325, rue de l'Université, Québec, QC G1V 0A6, Canada
Istituto di Chimica e Tecnologia Dei Polimeri, CNR, Via P. Gaifami, 18, 95126 Catania, Italy
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Synthesis, chemical characterization and biological activity of new histone acetylation/deacetylation specific inhibitors: A novel and potential approach to cancer therapy
Synthesis, chemical characterization and biological activity of new histone acetylation/deacetylation specific inhibitors: A novel and potential approach to cancer therapy
No results.
Synthesis, chemical characterization and biological activity of new histone acetylation/deacetylation specific inhibitors: A novel and potential approach to cancer therapy
Petraglia F, Singh AA, Carafa V, Nebbioso A, Conte M, Scisciola L, Valente S, Baldi A, Mandoli A, Petrizzi VB, Ingenito C, De Falco S, Cicatiello V, Apicella I, Janssen-megens EM, Kim B, Yi G, Logie C, Heath S, Ruvo M, Wierenga ATJ, Flicek P, Yaspo ML, Della Valle V, Bernard O, Tomassi S, Novellino E, Feoli A, Sbardella G, Gut I, Vellenga E, Stunnenberg HG, Mai A, Martens JHA, Altucci L * Combined HAT/EZH2 modulation leads to cancer-selective cell death(284 views) Oncotarget (ISSN: 1949-2553electronic, 1949-2553linking), 2018 May 22; 9(39): 25630-25646. Impact Factor:5.008 ViewExport to BibTeXExport to EndNote