Discovery Of Small Peptide Antagonists Of Ped/Pea15-D4alpha Interaction From Simplified Combinatorial Libraries(480 views) Scognamiglio PL, Doti N, Grieco P, Pedone C, Ruvo M, Marasco D
Chem Biol Drug Des (ISSN: 1747-0277, 1747-0285), 2011 May; 77(5): 319-327.
Department of Biological Sciences, School of Biotechnological Sciences, University of Naples Federico II, Via Mezzocannone, 16, 80134, Naples, Italy
Department of Pharmaceutical and Toxicological Chemistry, University of Naples ''Federico II'', Via Montesano 49, Naples, Italy
Institute of Biostructures and Bioimaging - CNR, Via Mezzocannone 16, 80134, Naples, Italy
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Balakin, K. V., Kozintsev, A. V., Kiselyov, A. S., Savchuk, N. P., Rational design approaches to chemical libraries for hit identification (2006) Curr Drug Discov Technol, 3, pp. 49-65
Ecker, D. J., Crooke, S. T., Combinatorial drug discovery: which methods will produce the greatest value? (1995) Biotechnology (NY), 13, pp. 351-360
Kennedy, J. P., Williams, L., Bridges, T. M., Daniels, R. N., Weaver, D., Lindsley, C. W., Application of combinatorial chemistry science on modern drug discovery (2008) J Comb Chem, 10, pp. 345-354
Wells, J. A., McClendon, C. L., Reaching for high-hanging fruit in drug discovery at protein-protein interfaces (2007) Nature, 450, pp. 1001-1009
Shultz, M. D., Ham, Y. W., Lee, S. G., Davis, D. A., Brown, C., Chmielewski, J., Small-molecule dimerization inhibitors of wild-type and mutant HIV protease: a focused library approach (2004) J Am Chem Soc, 126, pp. 9886-9887
Zhao, H. F., Kiyota, T., Chowdhury, S., Purisima, E., Banville, D., Konishi, Y., Shen, S. H., A mammalian genetic system to screen for small molecules capable of disrupting protein-protein interactions (2004) Anal Chem, 76, pp. 2922-2927
Sillerud, L. O., Larson, R. S., Design and structure of peptide and peptidomimetic antagonists of protein-protein interaction (2005) Curr Protein Pept Sci, 6, pp. 151-169
Martin, E. J., Blaney, J. M., Siani, M. A., Spellmeyer, D. C., Wong, A. K., Moos, W. H., Measuring diversity: experimental design of combinatorial libraries for drug discovery (1995) J Med Chem, 38, pp. 1431-1436
Fields, G. B., Noble, R. L., Solid phase peptide synthesis utilizing 9-fluorenylmethoxycarbonyl amino acids (1990) Int J Pept Protein Res, 35, pp. 161-214
Geysen, H. M., Rodda, S. J., Mason, T. J., A priori delineation of a peptide which mimics a discontinuous antigenic determinant (1986) Mol Immunol, 23, pp. 709-715
Flier, J. S., Insulin receptors and insulin resistance (1983) Annu Rev Med, 34, pp. 145-160
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Arkin, M. R., Randal, M., DeLano, W. L., Hyde, J., Luong, T. N., Oslob, J. D., Raphael, D. R., Braisted, A. C., Binding of small molecules to an adaptive protein-protein interface (2003) Proc Natl Acad Sci USA, 100, pp. 1603-1608
Sidhu, S. S., Fairbrother, W. J., Deshayes, K., Exploring protein-protein interactions with phage display (2003) Chembiochem, 4, pp. 14-25
Pillutla, R. C., Hsiao, K. C., Beasley, J. R., Brandt, J., Ostergaard, S., Hansen, P. H., Spetzler, J. C., Goldstein, N. I., Peptides identify the critical hotspots involved in the biological activation of the insulin receptor (2002) J Biol Chem, 277, pp. 22590-22594
Nakamura, G. R., Reynolds, M. E., Chen, Y. M., Starovasnik, M. A., Lowman, H. B., Stable "zeta" peptides that act as potent antagonists of the high-affinity IgE receptor (2002) Proc Natl Acad Sci USA, 99, pp. 1303-1308
Besterman, J. M., Duronio, V., Cuatrecasas, P., Rapid formation of diacylglycerol from phosphatidylcholine: a pathway for generation of a second messenger (1986) Proc Natl Acad Sci USA, 83, pp. 6785-6789
Sung, T. C., Zhang, Y., Morris, A. J., Frohman, M. A., Structural analysis of human phospholipase D1 (1999) J Biol Chem, 274, pp. 3659-3666
Xie, Z., Ho, W. T., Exton, J., Association of the N- and C-terminal domains of Phospholipase D is required for catalytic activity (1998) J Biol Chem, 273, pp. 34679-34682
Discovery Of Small Peptide Antagonists Of Ped/Pea15-D4alpha Interaction From Simplified Combinatorial Libraries
Vitiello M, Finamore E, Falanga A, Raieta K, Cantisani M, Galdiero F, Pedone C, Galdiero M, Galdiero S * Fusion in Coq(479 views) Lecture Notes In Computer Science (ISSN: 0302-9743, 0302-974335404636319783540463634, 0302-974335402975459783540297543), 2001; 2178LNCS: 583-596. Impact Factor:0.415 ViewExport to BibTeXExport to EndNote