High-Throughput Screening (HTS) by NMR Guided Identification of Novel Agents Targeting the Protein Docking Domain of YopH(422 views) Bottini A, Wu B, Barile E, De SK, Leone M, Pellecchia M
Chemmedchem (ISSN: 1860-7179, 1860-7187, 1860-7179linking), 2015 Nov 23; 11(8): 919-927.
Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, CA, 92037 (USA)., Sanford Burnham Prebys Graduate School of Biomedical Sciences, 10901 North Torrey Pines Road, La Jolla, CA, 92037 (USA)., Division of Biomedical Sciences, School of Medicine, University of California Riverside, 900 University Avenue, Riverside, CA, 92521 (USA)., Institute of Biostructures & Bioimaging, National Research Council (IBB-CNR), Via De Amicis 95, Naples, 80145 (Italy)., Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, CA, 92037 (USA). maurizio.pellecchia@ucr.edu., Division of Biomedical Sciences, School of Medicine, University of California Riverside, 900 University Avenue, Riverside, CA, 92521 (USA). maurizio.pellecchia@ucr.edu.,
1. Sanford Burnham Prebys Medical Discovery Institute, 10901 North Torrey Pines Road, La Jolla, CA, 92037 (USA
References: Baell, J.B., Holloway, G.A., (2010) J. Med. Chem., 53, pp. 2719-274
Baell, J., Walters, M.A., (2014) Nature, 513, pp. 481-483
Erlanson, D.A., McDowell, R.S., O'Brien, T., (2004) J. Med. Chem., 47, pp. 3463-3482
Bauman, J.D., Patel, D., Arnold, E., (2011) Top. Curr. Chem., 317, pp. 181-200
Visegrády, A., Keseru, G.M., (2013) Expert Opin. Drug Discovery, 8, pp. 811-820
Barile, E., Pellecchia, M., (2014) Chem. Rev., 114, pp. 4749-4763
Pellecchia, M., Bertini, I., Cowburn, D., Dalvit, C., Giralt, E., Jahnke, W., James, T.L., Siegal, G., (2008) Nat. Rev. Drug Discovery, 7, pp. 738-745
Pellecchia, M., (2005) Chem. Biol., 12, pp. 961-971
Pellecchia, M., Becattini, B., Crowell, K.J., Fattorusso, R., Forino, M., Fragai, M., Jung, D., Tautz, L., (2004) Expert Opin. Ther. Targets, 8, pp. 597-611
Wu, B., Barile, E., De, S.K., Wei, J., Purves, A., Pellecchia, M., (2015) Curr. Top. Med. Chem., 15, pp. 2032-2042
Pellecchia, M., Sem, D.S., Wuthrich, K., (2002) Nat. Rev. Drug Discovery, 1, pp. 211-219
Wu, B., Zhang, Z., Noberini, R., Barile, E., Giulianotti, M., Pinilla, C., Houghten, R.A., Pellecchia, M., (2013) Chem. Biol., 20, pp. 19-33