Epigenetic modulation of mGlu2 receptors by histone deacetylase inhibitors in the treatment of inflammatory pain(497 views) Chiechio S, Zammataro M, Morales ME, Busceti CL, Drago F, Th Gereau RW, Copani A, Nicoletti F
Department of Pharmaceutical Sciences, University of Catania, Italy
Department of Experimental and Clinical Pharmacology, University of Catania, Italy
Washington University Pain Center, Department of Anesthesiology, Washington University School of Medicine, St. Louis, MO, United States
Department of Human Physiology and Pharmacology, University of Rome, La Sapienza, Italy
I.B.B., CNR-Catania, Italy
I.N.M. Neuromed., Pozzilli, Italy
I. B. B., CNR-Catania, Italy
I. N. M. Neuromed., Pozzilli, Italy
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Ashburner, B. P., Westerheide, S. D., Baldwin Jr., A. S., The p65 (RelA) subunit of NF-kappaB interacts with the histone deacetylase (HDAC) corepressors HDAC1 and HDAC2 to negatively regulate gene expression (2001) Molecular and Cellular Biology, 21 (20), pp. 7065-7077. , DOI 10. 1128/MCB. 21. 20. 7065-7077. 200
Carlton, S. M., Hargett, G. L., Coggeshall, R. E., Localization of metabotropic glutamate receptors 2/3 on primary afferent axons in the rat (2001) Neuroscience, 105 (4), pp. 957-969. , DOI 10. 1016/S0306-4522 (01) 00238-X, PII S030645220100238X
Chen, L. -F., Fischle, W., Verdin, E., Greene, W. C., Duration of nuclear NF-kappaB action regulated by reversible acetylation (2001) Science, 293 (5535), pp. 1653-1657. , DOI 10. 1126/science. 1062374
Chen, L. F., Greene, W. C., Shaping the nuclear action of NF-kappaB (2004) Nat Rev Mol Cell Biol, 5, pp. 392-401
Chen, L. -F., Mu, Y., Greene, W. C., Acetylation of RelA at discrete sites regulates distinct nuclear functions of NF-kappaB (2002) EMBO Journal, 21 (23), pp. 6539-6548. , DOI 10. 1093/emboj/cdf660
Coderre, T. J., Contribution of protein kinase C to central sensitization and persistent pain following tissue injury (1992) Neurosci Lett, 140, pp. 181-184
Coderre, T. J., Melzack, R., The contribution of excitatory amino acids to central sensitization and persistent nociception after formalin-induced tissue injury (1992) J Neurosci, 12, pp. 3665-3670
Dougherty, P. M., Cata, J. P., Cordella, J. V., Burton, A., Weng, H. -R., Taxol-induced sensory disturbance is characterized by preferential impairment of myelinated fiber function in cancer patients (2004) Pain, 109 (1-2), pp. 132-142. , DOI 10. 1016/j. pain. 2004. 01. 021, PII S0304395904000533
Fundytus, M. E., Glutamate receptors and nociception: Implications for the drug treatment of pain (2001) CNS Drugs, 15 (1), pp. 29-58
Jones, C. K., Eberle, E. L., Peters, S. C., Monn, J. A., Shannon, H. E., Analgesic effects of the selective group II (mGlu2/3) metabotropic glutamate receptor agonists LY379268 and LY389795 in persistent and inflammatory pain models after acute and repeated dosing (2005) Neuropharmacology, 49 (SUPPL.), pp. 206-218. , DOI 10. 1016/j. neuropharm. 2005. 05. 008, PII S0028390805001899
Lin, Y. C., Flock, K. E., Cook, R. J., Hunkele, A. J., Loh, H. H., Ko, J. L., Effects of trichostatin a on neuronal mu-opioid receptor gene expression (2008) Brain Res, 1246, pp. 1-10
Malmberg, A. B., Gilbert, H., McCabe, R. T., Basbaum, A. I., Powerful antinociceptive effects of the cone snail venom-derived subtype-selective NMDA receptor antagonists conantokins G and T (2003) Pain, 101 (1-2), pp. 109-116. , DOI 10. 1016/S0304-3959 (02) 00303-2
Patil, S. T., Zhang, L., Martenyi, F., Lowe, S. L., Jackson, K. A., Andreev, B. V., Avedisova, A. S., Schoepp, D. D., Activation of mGlu2/3 receptors as a new approach to treat schizophrenia: A randomized Phase 2 clinical trial (2007) Nature Medicine, 13 (9), pp. 1102-1107. , DOI 10. 1038/nm1632, PII NM1632
Polomano, R. C., Mannes, A. J., Clark, U. S., Bennett, G. J., A painful peripheral neuropathy in the rat produced by the chemotherapeutic drug, paclitaxel (2001) Pain, 94 (3), pp. 293-304. , DOI 10. 1016/S0304-3959 (01) 00363-3, PII S0304395901003633
Schoepp, D. D., Jane, D. E., Monn, J. A., Pharmacological agents acting at subtypes of metabotropic glutamate receptors (1999) Neuropharmacology, 38 (10), pp. 1431-1476. , DOI 10. 1016/S0028-3908 (99) 00092-1, PII S0028390899000921
Simmons, R. M., Webster, A. A., Kalra, A. B., Iyengar, S., Group II mGluR receptor agonists are effective in persistent and neuropathic pain models in rats (2002) Pharmacol Biochem Behav, 73, pp. 419-427
Strahl, B. D., Allis, C. D., The language of covalent histone modifications (2000) Nature, 403 (6765), pp. 41-45. , DOI 10. 1038/47412
Tj lsen, A., Berge, O. G., Hunskaar, S., Rosland, J. H., Hole, K., The formalin test: An evaluation of the method (1992) Pain, 51, pp. 5-17
Xu, W. S., Parmigiani, R. B., Marks, P. A., Histone deacetylase inhibitors: Molecular mechanisms of action (2007) Oncogene, 26 (37), pp. 5541-5552. , DOI 10. 1038/sj. onc. 1210620, PII 1210620
Yang, X. -J., Seto, E., HATs and HDACs: From structure, function and regulation to novel strategies for therapy and prevention (2007) Oncogene, 26 (37), pp. 5310-5318. , DOI 10. 1038/sj. onc. 1210599, PII 1210599
Epigenetic modulation of mGlu2 receptors by histone deacetylase inhibitors in the treatment of inflammatory pain
Vitiello M, Finamore E, Falanga A, Raieta K, Cantisani M, Galdiero F, Pedone C, Galdiero M, Galdiero S * Fusion in Coq(479 views) Lecture Notes In Computer Science (ISSN: 0302-9743, 0302-974335404636319783540463634, 0302-974335402975459783540297543), 2001; 2178LNCS: 583-596. Impact Factor:0.415 ViewExport to BibTeXExport to EndNote