In vitro autoradiography and in vivo evaluation in cynomolgus monkey of [18F]FE-PE2I, a new dopamine transporter PET radioligand(1515 views) Varrone A, Steiger C, Schou M, Takano A, Finnema SJ, Guilloteau D, Gulyas B, Halldin C
Keywords: Dopamine Transporter (dat), Kinetics, Metabolism, Midbrain, Substantia Nigra, [2 Beta Carbomethoxy 3 Beta (4 Fluorophenyl) 8 (2 Fluoroethyl) Nortropane] F 18, Beta Carboxymethoxy 3 Beta (4 Iodophenyltropane), Citalopram, Maprotiline, Radioligand, Tracer, Unclassified Drug, Vanoxerine, Animal Experiment, Animal Tissue, Article, Autoradiography, Caudate Nucleus, Cerebellum, Controlled Study, Corpus Striatum, Drug Binding, Drug Elimination, Drug Metabolism, Drug Uptake, Human, Human Tissue, In Vitro Study, In Vivo Study, Ligand Binding, Mesencephalon, Methodology, Monkey, Neocortex, Nonhuman, Positron Emission Tomography, Priority Journal, Putamen, Quantitative Analysis, Rodent, Thalamus, Competitive, Dopamine Plasma Membrane Transport Proteins, Dopamine Uptake Inhibitors, Dose-Response Relationship, Macaca Fascicularis, Metabolic Clearance Rate, Piperazines, Positron-Emission Tomography, Postmortem Changes, Protein Binding, Radiopharmaceuticals, Serotonin Uptake Inhibitors, Tissue Distribution,
Affiliations: *** IBB - CNR ***
Karolinska Institutet, Department of Clinical Neuroscience, Karolinska Hospital, SE-17176, Stockholm, Sweden
Stockholm Brain Institute, Stockholm, Sweden
Inserm U930, Université François Rabelais de Tours, Tours, France
Medicinal Chemistry AstraZeneca R and D, Södertäljie, Sweden
References: Not available.
In vitro autoradiography and in vivo evaluation in cynomolgus monkey of [18F]FE-PE2I, a new dopamine transporter PET radioligand
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